Chuang, Shang-Ju

6-Thioguanine is a noncompetitive and slow binding inhibitor of human deubiquitinating protease USP2. [electronic resource] - Scientific reports 02 2018 - 3102 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

2045-2322

10.1038/s41598-018-21476-w doi


Crystallography, X-Ray--methods
Deubiquitinating Enzymes--antagonists & inhibitors
Endopeptidases--metabolism
Humans
Kinetics
Protein Processing, Post-Translational
Thioguanine--metabolism
Ubiquitin Thiolesterase
Ubiquitination--physiology