Zhang, Ning
Host-parasite co-metabolic activation of antitrypanosomal aminomethyl-benzoxaboroles. [electronic resource]
- PLoS pathogens 02 2018
- e1006850 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
1553-7374
10.1371/journal.ppat.1006850 doi
Activation, Metabolic
Aldehyde Dehydrogenase--antagonists & inhibitors
Aldehyde Oxidoreductases--antagonists & inhibitors
Amine Oxidase (Copper-Containing)--antagonists & inhibitors
Amino Acid Substitution
Animals
Boron Compounds--chemistry
Drug Resistance
High-Throughput Screening Assays
Humans
Models, Biological
Molecular Structure
Mutation
Phylogeny
Prodrugs--chemistry
Protein Interaction Domains and Motifs
RNA Interference
Rats
Recombinant Fusion Proteins--chemistry
Recombinant Proteins--chemistry
Structure-Activity Relationship
Trypanocidal Agents--chemistry
Trypanosoma brucei brucei--drug effects