TY  - GEN
AU  - Korepanova,Alla
AU  - Longenecker,Kenton L
AU  - Pratt,Steve D
AU  - Panchal,Sanjay C
AU  - Clark,Richard F
AU  - Lake,Marc
AU  - Gopalakrishnan,Sujatha M
AU  - Raich,Diana
AU  - Sun,Chaohong
AU  - Petros,Andrew M
TI  - Fragment-based discovery of a potent NAMPT inhibitor
SN  - 1464-3405
PY  - 2019///0530
KW  - Acrylamides
KW  - chemical synthesis
KW  - Cytokines
KW  - antagonists & inhibitors
KW  - Dose-Response Relationship, Drug
KW  - Drug Discovery
KW  - Drug Evaluation, Preclinical
KW  - Enzyme Inhibitors
KW  - Fluorescence Resonance Energy Transfer
KW  - Humans
KW  - Molecular Docking Simulation
KW  - Molecular Structure
KW  - Nicotinamide Phosphoribosyltransferase
KW  - Piperidines
KW  - Structure-Activity Relationship
N1  - Publication Type: Journal Article; Research Support, U.S. Gov't, Non-P.H.S
UR  - https://doi.org/10.1016/j.bmcl.2017.12.023
ER  -