Korepanova, Alla
Fragment-based discovery of a potent NAMPT inhibitor. [electronic resource]
- Bioorganic & medicinal chemistry letters 02 2018
- 437-440 p. digital
Publication Type: Journal Article; Research Support, U.S. Gov't, Non-P.H.S.
1464-3405
10.1016/j.bmcl.2017.12.023 doi
Acrylamides--chemical synthesis
Cytokines--antagonists & inhibitors
Dose-Response Relationship, Drug
Drug Discovery
Drug Evaluation, Preclinical
Enzyme Inhibitors--chemical synthesis
Fluorescence Resonance Energy Transfer
Humans
Molecular Docking Simulation
Molecular Structure
Nicotinamide Phosphoribosyltransferase--antagonists & inhibitors
Piperidines--chemical synthesis
Structure-Activity Relationship