Korepanova, Alla

Fragment-based discovery of a potent NAMPT inhibitor. [electronic resource] - Bioorganic & medicinal chemistry letters 02 2018 - 437-440 p. digital

Publication Type: Journal Article; Research Support, U.S. Gov't, Non-P.H.S.

1464-3405

10.1016/j.bmcl.2017.12.023 doi


Acrylamides--chemical synthesis
Cytokines--antagonists & inhibitors
Dose-Response Relationship, Drug
Drug Discovery
Drug Evaluation, Preclinical
Enzyme Inhibitors--chemical synthesis
Fluorescence Resonance Energy Transfer
Humans
Molecular Docking Simulation
Molecular Structure
Nicotinamide Phosphoribosyltransferase--antagonists & inhibitors
Piperidines--chemical synthesis
Structure-Activity Relationship