Drug-induced inhibition of phosphorylation of STAT5 overrides drug resistance in neoplastic mast cells. [electronic resource]
- Leukemia 04 2018
- 1016-1022 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1476-5551
10.1038/leu.2017.338 doi
Adult Aged Aged, 80 and over Animals Apoptosis--drug effects Cell Cycle Checkpoints--drug effects Cell Line, Tumor Dasatinib--pharmacology Dogs Drug Resistance, Neoplasm--drug effects Drug Synergism Female G2 Phase Cell Cycle Checkpoints--drug effects Humans Leukemia, Mast-Cell--drug therapy Male Mast Cells--drug effects Mastocytosis, Systemic--drug therapy Middle Aged Norbornanes--pharmacology Phosphorylation--drug effects Protein Kinase Inhibitors--pharmacology Proto-Oncogene Proteins c-kit--metabolism Pyrimidines--pharmacology STAT5 Transcription Factor--metabolism Staurosporine--analogs & derivatives Tumor Suppressor Proteins--metabolism Young Adult