Peter, B

Drug-induced inhibition of phosphorylation of STAT5 overrides drug resistance in neoplastic mast cells. [electronic resource] - Leukemia 04 2018 - 1016-1022 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1476-5551

10.1038/leu.2017.338 doi


Adult
Aged
Aged, 80 and over
Animals
Apoptosis--drug effects
Cell Cycle Checkpoints--drug effects
Cell Line, Tumor
Dasatinib--pharmacology
Dogs
Drug Resistance, Neoplasm--drug effects
Drug Synergism
Female
G2 Phase Cell Cycle Checkpoints--drug effects
Humans
Leukemia, Mast-Cell--drug therapy
Male
Mast Cells--drug effects
Mastocytosis, Systemic--drug therapy
Middle Aged
Norbornanes--pharmacology
Phosphorylation--drug effects
Protein Kinase Inhibitors--pharmacology
Proto-Oncogene Proteins c-kit--metabolism
Pyrimidines--pharmacology
STAT5 Transcription Factor--metabolism
Staurosporine--analogs & derivatives
Tumor Suppressor Proteins--metabolism
Young Adult