Discovery of LY3104607: A Potent and Selective G Protein-Coupled Receptor 40 (GPR40) Agonist with Optimized Pharmacokinetic Properties to Support Once Daily Oral Treatment in Patients with Type 2 Diabetes Mellitus. [electronic resource]
- Journal of medicinal chemistry 02 2018
- 934-945 p. digital
Publication Type: Journal Article
1520-4804
10.1021/acs.jmedchem.7b01411 doi
Administration, Oral Animals Diabetes Mellitus, Type 2--drug therapy Dogs Drug Discovery Humans Hypoglycemic Agents--administration & dosage Male Pyridines--administration & dosage Rats Receptors, G-Protein-Coupled--agonists Structure-Activity Relationship Triazoles--administration & dosage