Hamdouchi, Chafiq

Discovery of LY3104607: A Potent and Selective G Protein-Coupled Receptor 40 (GPR40) Agonist with Optimized Pharmacokinetic Properties to Support Once Daily Oral Treatment in Patients with Type 2 Diabetes Mellitus. [electronic resource] - Journal of medicinal chemistry 02 2018 - 934-945 p. digital

Publication Type: Journal Article

1520-4804

10.1021/acs.jmedchem.7b01411 doi


Administration, Oral
Animals
Diabetes Mellitus, Type 2--drug therapy
Dogs
Drug Discovery
Humans
Hypoglycemic Agents--administration & dosage
Male
Pyridines--administration & dosage
Rats
Receptors, G-Protein-Coupled--agonists
Structure-Activity Relationship
Triazoles--administration & dosage