Lis, Christian

Development of Erasin: a chromone-based STAT3 inhibitor which induces apoptosis in Erlotinib-resistant lung cancer cells. [electronic resource] - Scientific reports 12 2017 - 17390 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.

2045-2322

10.1038/s41598-017-17600-x doi


Antineoplastic Agents--pharmacology
Apoptosis--drug effects
Carcinoma, Non-Small-Cell Lung--drug therapy
Cell Line, Tumor
Chromones--pharmacology
Humans
Lung Neoplasms--drug therapy
Molecular Docking Simulation
Phosphorylation
Protein Processing, Post-Translational
STAT1 Transcription Factor--antagonists & inhibitors
STAT3 Transcription Factor--antagonists & inhibitors
STAT5 Transcription Factor--antagonists & inhibitors
Structure-Activity Relationship
Tumor Suppressor Proteins--antagonists & inhibitors
src Homology Domains