Morishita, Ko Novel Non-carboxylate Benzoylsulfonamide-Based Protein Tyrosine Phosphatase 1B Inhibitors with Non-competitive Actions. [electronic resource] - Chemical & pharmaceutical bulletin 2017 - 1144-1160 p. digital Publication Type: Journal Article ISSN: 1347-5223 Standard No.: 10.1248/cpb.c17-00635 doi Subjects--Topical Terms: Administration, OralAllosteric Regulation--drug effectsAmino Acid SequenceAnimalsBinding SitesBlood Glucose--analysisDogsEnzyme Inhibitors--chemistryHypoglycemic Agents--chemistryInhibitory Concentration 50MaleMiceMice, ObeseMolecular Dynamics SimulationProtein Tyrosine Phosphatase, Non-Receptor Type 1--antagonists & inhibitorsRatsRats, Sprague-DawleySequence AlignmentStructure-Activity RelationshipSulfonamides--chemistry