Morishita, Ko

Novel Non-carboxylate Benzoylsulfonamide-Based Protein Tyrosine Phosphatase 1B Inhibitors with Non-competitive Actions. [electronic resource] - Chemical & pharmaceutical bulletin 2017 - 1144-1160 p. digital

Publication Type: Journal Article

1347-5223

10.1248/cpb.c17-00635 doi


Administration, Oral
Allosteric Regulation--drug effects
Amino Acid Sequence
Animals
Binding Sites
Blood Glucose--analysis
Dogs
Enzyme Inhibitors--chemistry
Hypoglycemic Agents--chemistry
Inhibitory Concentration 50
Male
Mice
Mice, Obese
Molecular Dynamics Simulation
Protein Tyrosine Phosphatase, Non-Receptor Type 1--antagonists & inhibitors
Rats
Rats, Sprague-Dawley
Sequence Alignment
Structure-Activity Relationship
Sulfonamides--chemistry