Loudon, Peter

Demonstration of an anti-hyperalgesic effect of a novel pan-Trk inhibitor PF-06273340 in a battery of human evoked pain models. [electronic resource] - British journal of clinical pharmacology 02 2018 - 301-309 p. digital

Publication Type: Journal Article; Randomized Controlled Trial; Research Support, Non-U.S. Gov't

1365-2125

10.1111/bcp.13448 doi


Adolescent
Adult
Analgesics--administration & dosage
Cross-Over Studies
Dose-Response Relationship, Drug
Double-Blind Method
Healthy Volunteers
Humans
Hyperalgesia--drug therapy
Male
Membrane Glycoproteins--antagonists & inhibitors
Middle Aged
Pain Threshold--drug effects
Pyrimidines--administration & dosage
Pyrroles--administration & dosage
Receptor, trkA--antagonists & inhibitors
Receptor, trkB--antagonists & inhibitors
Receptor, trkC--antagonists & inhibitors
Young Adult