Murray, Michael

Variation in the Response of Clozapine Biotransformation Pathways in Human Hepatic Microsomes to CYP1A2- and CYP3A4-selective Inhibitors. [electronic resource] - Basic & clinical pharmacology & toxicology Apr 2018 - 388-395 p. digital

Publication Type: Journal Article

1742-7843

10.1111/bcpt.12933 doi


Antipsychotic Agents--metabolism
Biotransformation
Clozapine--analogs & derivatives
Cytochrome P-450 CYP1A2--metabolism
Cytochrome P-450 CYP1A2 Inhibitors--pharmacology
Cytochrome P-450 CYP3A--metabolism
Cytochrome P-450 CYP3A Inhibitors--pharmacology
Drug Interactions
Fluvoxamine--pharmacology
Humans
Hydroxylation
Ketoconazole--pharmacology
Liver--cytology
Microsomes, Liver--drug effects
Oxidation-Reduction