Colas, Claire
Chemical Modulation of the Human Oligopeptide Transporter 1, hPepT1. [electronic resource]
- Molecular pharmaceutics 12 2017
- 4685-4693 p. digital
Publication Type: Journal Article; Research Support, U.S. Gov't, Non-P.H.S.; Research Support, N.I.H., Extramural
1543-8392
10.1021/acs.molpharmaceut.7b00775 doi
Biological Transport, Active--drug effects
Drug Evaluation, Preclinical--methods
Humans
Inhibitory Concentration 50
Intestinal Absorption--drug effects
Kinetics
Ligands
Models, Chemical
Models, Molecular
Molecular Docking Simulation
Oligopeptides--chemistry
Peptide Transporter 1--antagonists & inhibitors
Prodrugs--chemistry