TY - GEN AU - Asquith,Christopher R M AU - Laitinen,Tuomo AU - Bennett,James M AU - Godoi,Paulo H AU - East,Michael P AU - Tizzard,Graham J AU - Graves,Lee M AU - Johnson,Gary L AU - Dornsife,Ronna E AU - Wells,Carrow I AU - Elkins,Jonathan M AU - Willson,Timothy M AU - Zuercher,William J TI - Identification and Optimization of 4-Anilinoquinolines as Inhibitors of Cyclin G Associated Kinase SN - 1860-7187 PY - 2018///1004 KW - Aniline Compounds KW - chemistry KW - Binding Sites KW - Catalytic Domain KW - Drug Design KW - Endocytosis KW - drug effects KW - Humans KW - Intracellular Signaling Peptides and Proteins KW - antagonists & inhibitors KW - Kinetics KW - Molecular Docking Simulation KW - Protein Binding KW - Protein Kinase Inhibitors KW - Protein Serine-Threonine Kinases KW - Quinazolines KW - Structure-Activity Relationship KW - Viruses KW - pathogenicity N1 - Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't UR - https://doi.org/10.1002/cmdc.201700663 ER -