Identification and Optimization of 4-Anilinoquinolines as Inhibitors of Cyclin G Associated Kinase. [electronic resource]
- ChemMedChem 01 2018
- 48-66 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1860-7187
10.1002/cmdc.201700663 doi
Aniline Compounds--chemistry Binding Sites Catalytic Domain Drug Design Endocytosis--drug effects Humans Intracellular Signaling Peptides and Proteins--antagonists & inhibitors Kinetics Molecular Docking Simulation Protein Binding Protein Kinase Inhibitors--chemistry Protein Serine-Threonine Kinases--antagonists & inhibitors Quinazolines--chemistry Structure-Activity Relationship Viruses--pathogenicity