TY  - GEN
AU  - Bouley,Renee
AU  - Waldschmidt,Helen V
AU  - Cato,M Claire
AU  - Cannavo,Alessandro
AU  - Song,Jianliang
AU  - Cheung,Joseph Y
AU  - Yao,Xin-Qiu
AU  - Koch,Walter J
AU  - Larsen,Scott D
AU  - Tesmer,John J G
TI  - Structural Determinants Influencing the Potency and Selectivity of Indazole-Paroxetine Hybrid G Protein-Coupled Receptor Kinase 2 Inhibitors
SN  - 1521-0111
PY  - 2017///1128
KW  - Animals
KW  - G-Protein-Coupled Receptor Kinase 2
KW  - antagonists & inhibitors
KW  - G-Protein-Coupled Receptor Kinase 5
KW  - pharmacology
KW  - Humans
KW  - Indazoles
KW  - Mice
KW  - Mice, Inbred C57BL
KW  - Models, Molecular
KW  - Paroxetine
KW  - Protein Kinase Inhibitors
KW  - Selective Serotonin Reuptake Inhibitors
KW  - rho-Associated Kinases
KW  - metabolism
N1  - Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S
UR  - https://doi.org/10.1124/mol.117.110130
ER  -