Bouley, Renee

Structural Determinants Influencing the Potency and Selectivity of Indazole-Paroxetine Hybrid G Protein-Coupled Receptor Kinase 2 Inhibitors. [electronic resource] - Molecular pharmacology 12 2017 - 707-717 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.

1521-0111

10.1124/mol.117.110130 doi


Animals
G-Protein-Coupled Receptor Kinase 2--antagonists & inhibitors
G-Protein-Coupled Receptor Kinase 5--pharmacology
Humans
Indazoles--pharmacology
Mice
Mice, Inbred C57BL
Models, Molecular
Paroxetine--pharmacology
Protein Kinase Inhibitors--pharmacology
Selective Serotonin Reuptake Inhibitors
rho-Associated Kinases--metabolism