Arnold, Michael A

4-Hydroxy-2-pyridones: Discovery and evaluation of a novel class of antibacterial agents targeting DNA synthesis. [electronic resource] - Bioorganic & medicinal chemistry letters 11 2017 - 5014-5021 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2017.10.006 doi


Animals
Anti-Bacterial Agents--chemistry
Azabicyclo Compounds--chemistry
DNA--chemistry
Drug Evaluation, Preclinical
Escherichia coli--drug effects
Gram-Negative Bacteria--drug effects
Gram-Negative Bacterial Infections--drug therapy
Half-Life
Mice
Microbial Sensitivity Tests
Niacin--analogs & derivatives
Pyridines--chemistry
Structure-Activity Relationship