Arnold, Michael A 4-Hydroxy-2-pyridones: Discovery and evaluation of a novel class of antibacterial agents targeting DNA synthesis. [electronic resource] - Bioorganic & medicinal chemistry letters 11 2017 - 5014-5021 p. digital Publication Type: Journal Article ISSN: 1464-3405 Standard No.: 10.1016/j.bmcl.2017.10.006 doi Subjects--Topical Terms: AnimalsAnti-Bacterial Agents--chemistryAzabicyclo Compounds--chemistryDNA--chemistryDrug Evaluation, PreclinicalEscherichia coli--drug effectsGram-Negative Bacteria--drug effectsGram-Negative Bacterial Infections--drug therapyHalf-LifeMiceMicrobial Sensitivity TestsNiacin--analogs & derivativesPyridines--chemistryStructure-Activity Relationship