Simultaneous determination of a novel c-Met/AXL dual-target small-molecule inhibitor BPI-9016M and its metabolites in human plasma by liquid chromatography-tandem mass spectrometry: Application in a pharmacokinetic study in Chinese advanced solid tumor patients. [electronic resource]
- Journal of chromatography. B, Analytical technologies in the biomedical and life sciences Nov 2017
- 33-40 p. digital
Publication Type: Journal Article
1873-376X
10.1016/j.jchromb.2017.10.017 doi
Antineoplastic Agents--therapeutic use Chromatography, Liquid--methods Drug Stability Humans Linear Models Neoplasms--drug therapy Protein Kinase Inhibitors--therapeutic use Proto-Oncogene Proteins--antagonists & inhibitors Proto-Oncogene Proteins c-met--antagonists & inhibitors Receptor Protein-Tyrosine Kinases--antagonists & inhibitors Reproducibility of Results Sensitivity and Specificity Tandem Mass Spectrometry--methods Axl Receptor Tyrosine Kinase