Ponnusamy, Suriyan

Novel Selective Agents for the Degradation of Androgen Receptor Variants to Treat Castration-Resistant Prostate Cancer. [electronic resource] - Cancer research 11 2017 - 6282-6298 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1538-7445

10.1158/0008-5472.CAN-17-0976 doi


Alternative Splicing
Androgen Receptor Antagonists--chemistry
Anilides--chemistry
Animals
Cell Line, Tumor
Cell Proliferation--drug effects
Gene Expression Profiling--methods
Gene Expression Regulation, Neoplastic--drug effects
Humans
Indoles--chemistry
Male
Mice, Inbred NOD
Mice, Knockout
Mice, SCID
Molecular Structure
Prostatic Neoplasms, Castration-Resistant--drug therapy
Receptors, Androgen--genetics
Xenograft Model Antitumor Assays