Brägelmann, Johannes

Systematic Kinase Inhibitor Profiling Identifies CDK9 as a Synthetic Lethal Target in NUT Midline Carcinoma. [electronic resource] - Cell reports Sep 2017 - 2833-2845 p. digital

Publication Type: Journal Article

2211-1247

10.1016/j.celrep.2017.08.082 doi


Cell Cycle Proteins
Cell Line, Tumor
Cyclin T--metabolism
Cyclin-Dependent Kinase 9--antagonists & inhibitors
HEK293 Cells
High-Throughput Screening Assays
Humans
Molecular Targeted Therapy
Neoplasms--enzymology
Nuclear Proteins--antagonists & inhibitors
Protein Kinase Inhibitors--chemistry
RNA Polymerase II--metabolism
Transcription Elongation, Genetic--drug effects
Transcription Factors--antagonists & inhibitors
Transcription, Genetic--drug effects