Crivelli, Simone M

Synthesis, Radiosynthesis, and Preliminary in vitro and in vivo Evaluation of the Fluorinated Ceramide Trafficking Inhibitor (HPA-12) for Brain Applications. [electronic resource] - Journal of Alzheimer's disease : JAD 2017 - 783-794 p. digital

Publication Type: Journal Article

1875-8908

10.3233/JAD-161231 doi


Amides--chemical synthesis
Animals
Brain--diagnostic imaging
Ceramides--metabolism
Drug Evaluation, Preclinical
Drug Stability
Fluorine Radioisotopes
Halogenation
HeLa Cells
Humans
Male
Mice, Inbred C57BL
Microscopy, Fluorescence
Positron-Emission Tomography
Protein Serine-Threonine Kinases--metabolism
Radiopharmaceuticals--chemical synthesis