Synthesis, Radiosynthesis, and Preliminary in vitro and in vivo Evaluation of the Fluorinated Ceramide Trafficking Inhibitor (HPA-12) for Brain Applications. [electronic resource]
- Journal of Alzheimer's disease : JAD 2017
- 783-794 p. digital
Publication Type: Journal Article
1875-8908
10.3233/JAD-161231 doi
Amides--chemical synthesis Animals Brain--diagnostic imaging Ceramides--metabolism Drug Evaluation, Preclinical Drug Stability Fluorine Radioisotopes Halogenation HeLa Cells Humans Male Mice, Inbred C57BL Microscopy, Fluorescence Positron-Emission Tomography Protein Serine-Threonine Kinases--metabolism Radiopharmaceuticals--chemical synthesis