Song, Jia-Li

Design and synthesis of pregnenolone/2-cyanoacryloyl conjugates with dual NF-κB inhibitory and anti-proliferative activities. [electronic resource] - Bioorganic & medicinal chemistry letters 10 2017 - 4682-4686 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1464-3405

10.1016/j.bmcl.2017.09.013 doi


A549 Cells
Antineoplastic Agents--chemical synthesis
Cell Line, Tumor
Cell Proliferation--drug effects
Cell Survival--drug effects
Cyanoacrylates--chemistry
Drug Design
Drug Screening Assays, Antitumor
HL-60 Cells
Humans
MCF-7 Cells
NF-kappa B--antagonists & inhibitors
Pregnenolone--chemistry
Structure-Activity Relationship