SKLB188 inhibits the growth of head and neck squamous cell carcinoma by suppressing EGFR signalling. [electronic resource]
- British journal of cancer Oct 2017
- 1154-1163 p. digital
Publication Type: Journal Article
1532-1827
10.1038/bjc.2017.298 doi
Animals Apoptosis--drug effects Blotting, Western Carcinoma, Squamous Cell--metabolism Cell Proliferation--drug effects Cyclin A--drug effects Cyclin D1--drug effects Cyclin-Dependent Kinase 2--drug effects Cyclin-Dependent Kinase 4--drug effects Cyclin-Dependent Kinase Inhibitor p21--drug effects Cyclin-Dependent Kinase Inhibitor p27--drug effects Down-Regulation ErbB Receptors--antagonists & inhibitors G1 Phase Cell Cycle Checkpoints--drug effects Head and Neck Neoplasms--metabolism Humans Immunohistochemistry In Situ Nick-End Labeling In Vitro Techniques Mice Mice, Nude Molecular Docking Simulation Purines--pharmacology Signal Transduction Squamous Cell Carcinoma of Head and Neck Up-Regulation Xenograft Model Antitumor Assays cdc25 Phosphatases--drug effects