Discovery of Fragment-Derived Small Molecules for in Vivo Inhibition of Ketohexokinase (KHK). [electronic resource]
- Journal of medicinal chemistry 09 2017
- 7835-7849 p. digital
Publication Type: Journal Article; Research Support, U.S. Gov't, Non-P.H.S.
1520-4804
10.1021/acs.jmedchem.7b00947 doi
Animals Crystallography, X-Ray Drug Design Fructokinases--antagonists & inhibitors Humans Male Molecular Docking Simulation Protein Kinase Inhibitors--chemistry Pyridines--chemistry Rats Rats, Sprague-Dawley Small Molecule Libraries--chemistry