Huard, Kim

Discovery of Fragment-Derived Small Molecules for in Vivo Inhibition of Ketohexokinase (KHK). [electronic resource] - Journal of medicinal chemistry 09 2017 - 7835-7849 p. digital

Publication Type: Journal Article; Research Support, U.S. Gov't, Non-P.H.S.

1520-4804

10.1021/acs.jmedchem.7b00947 doi


Animals
Crystallography, X-Ray
Drug Design
Fructokinases--antagonists & inhibitors
Humans
Male
Molecular Docking Simulation
Protein Kinase Inhibitors--chemistry
Pyridines--chemistry
Rats
Rats, Sprague-Dawley
Small Molecule Libraries--chemistry