Ascites interferes with the activity of lurbinectedin and trabectedin: Potential role of their binding to alpha 1-acid glycoprotein. [electronic resource]
- Biochemical pharmacology 11 2017
- 52-62 p. digital
Publication Type: Journal Article
1873-2968
10.1016/j.bcp.2017.08.001 doi
Animals Antineoplastic Agents, Alkylating--metabolism Ascites--metabolism Carbolines--metabolism Cell Line, Tumor Dioxoles--metabolism Dose-Response Relationship, Drug Female Heterocyclic Compounds, 4 or More Rings--metabolism Humans Mice Mice, Nude Orosomucoid--metabolism Ovarian Neoplasms--drug therapy Protein Binding--physiology Tetrahydroisoquinolines--metabolism Trabectedin Tumor Cells, Cultured Xenograft Model Antitumor Assays--methods