Design, synthesis and biological evaluation of dual acetylcholinesterase and phosphodiesterase 5A inhibitors in treatment for Alzheimer's disease. [electronic resource]
- Bioorganic & medicinal chemistry letters 09 2017
- 4180-4184 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3405
10.1016/j.bmcl.2017.07.013 doi
Acetylcholinesterase--metabolism Alzheimer Disease--drug therapy Cell Line, Tumor Cell Survival--drug effects Cholinesterase Inhibitors--chemical synthesis Cyclic Nucleotide Phosphodiesterases, Type 5--metabolism Dose-Response Relationship, Drug Drug Design Humans Molecular Structure Phosphodiesterase Inhibitors--chemistry Structure-Activity Relationship