Joncour, Agnès

Discovery, Structure-Activity Relationship, and Binding Mode of an Imidazo[1,2-a]pyridine Series of Autotaxin Inhibitors. [electronic resource] - Journal of medicinal chemistry 09 2017 - 7371-7392 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1520-4804

10.1021/acs.jmedchem.7b00647 doi


Animals
Humans
Imidazoles--chemistry
Lysophosphatidylcholines--metabolism
Lysophospholipids--metabolism
Male
Mice
Molecular Docking Simulation
Phosphodiesterase Inhibitors--chemistry
Phosphoric Diester Hydrolases--chemistry
Pyridines--chemistry
Rats
Rats, Sprague-Dawley
Structure-Activity Relationship