TY  - GEN
AU  - González-Bacerio,Jorge
AU  - Maluf,Sarah El Chamy
AU  - Méndez,Yanira
AU  - Pascual,Isel
AU  - Florent,Isabelle
AU  - Melo,Pollyana M S
AU  - Budu,Alexandre
AU  - Ferreira,Juliana C
AU  - Moreno,Ernesto
AU  - Carmona,Adriana K
AU  - Rivera,Daniel G
AU  - Alonso Del Rivero,Maday
AU  - Gazarini,Marcos L
TI  - KBE009: An antimalarial bestatin-like inhibitor of the Plasmodium falciparum M1 aminopeptidase discovered in an Ugi multicomponent reaction-derived peptidomimetic library
SN  - 1464-3391
PY  - 2017///0926
KW  - Antimalarials
KW  - chemical synthesis
KW  - Binding Sites
KW  - CD13 Antigens
KW  - antagonists & inhibitors
KW  - Catalytic Domain
KW  - Cell Survival
KW  - drug effects
KW  - Dipeptides
KW  - Erythrocytes
KW  - cytology
KW  - Human Umbilical Vein Endothelial Cells
KW  - Humans
KW  - Leucine
KW  - analogs & derivatives
KW  - Molecular Docking Simulation
KW  - Peptidomimetics
KW  - Plasmodium falciparum
KW  - Protozoan Proteins
KW  - Recombinant Proteins
KW  - biosynthesis
KW  - Structure-Activity Relationship
N1  - Publication Type: Journal Article; Research Support, Non-U.S. Gov't
UR  - https://doi.org/10.1016/j.bmc.2017.06.047
ER  -