Tuning of β-glucosidase and α-galactosidase inhibition by generation and in situ screening of a library of pyrrolidine-triazole hybrid molecules. [electronic resource]
- European journal of medicinal chemistry Sep 2017
- 532-542 p. digital
Publication Type: Journal Article
1768-3254
10.1016/j.ejmech.2017.06.055 doi
Dose-Response Relationship, Drug Drug Evaluation, Preclinical Enzyme Inhibitors--chemical synthesis Humans Molecular Structure Pyrrolidines--chemical synthesis Small Molecule Libraries--chemical synthesis Structure-Activity Relationship Triazoles--chemical synthesis alpha-Galactosidase--antagonists & inhibitors beta-Glucosidase--antagonists & inhibitors