Martínez-Bailén, Macarena

Tuning of β-glucosidase and α-galactosidase inhibition by generation and in situ screening of a library of pyrrolidine-triazole hybrid molecules. [electronic resource] - European journal of medicinal chemistry Sep 2017 - 532-542 p. digital

Publication Type: Journal Article

1768-3254

10.1016/j.ejmech.2017.06.055 doi


Dose-Response Relationship, Drug
Drug Evaluation, Preclinical
Enzyme Inhibitors--chemical synthesis
Humans
Molecular Structure
Pyrrolidines--chemical synthesis
Small Molecule Libraries--chemical synthesis
Structure-Activity Relationship
Triazoles--chemical synthesis
alpha-Galactosidase--antagonists & inhibitors
beta-Glucosidase--antagonists & inhibitors