McConkey, Glenn A
Interconvertible geometric isomers of Plasmodium falciparum dihydroorotate dehydrogenase inhibitors exhibit multiple binding modes. [electronic resource]
- Bioorganic & medicinal chemistry letters 08 2017
- 3878-3882 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2017.06.052 doi
Acrylates--chemical synthesis
Dihydroorotate Dehydrogenase
Dose-Response Relationship, Drug
Molecular Docking Simulation
Molecular Structure
Oxidoreductases Acting on CH-CH Group Donors--antagonists & inhibitors
Plasmodium falciparum--enzymology
Structure-Activity Relationship