TY - GEN AU - Machaba,Kgothatso E AU - Mhlongo,Ndumiso N AU - Dokurugu,Yussif M AU - Soliman,Mahmoud Es TI - Tailored-pharmacophore model to enhance virtual screening and drug discovery: a case study on the identification of potential inhibitors against drug-resistant Mycobacterium tuberculosis (3R)-hydroxyacyl-ACP dehydratases SN - 1756-8927 PY - 2017///0912 KW - Drug Discovery KW - Drug Evaluation, Preclinical KW - Enoyl-CoA Hydratase KW - antagonists & inhibitors KW - Enzyme Inhibitors KW - chemical synthesis KW - Models, Molecular KW - Molecular Structure KW - Structure-Activity Relationship KW - Tuberculosis, Multidrug-Resistant KW - drug therapy N1 - Publication Type: Journal Article; Research Support, Non-U.S. Gov't UR - https://doi.org/10.4155/fmc-2017-0020 ER -