Mechanisms of Paradoxical Activation of AMPK by the Kinase Inhibitors SU6656 and Sorafenib. [electronic resource]
- Cell chemical biology Jul 2017
- 813-824.e4 p. digital
Publication Type: Journal Article
2451-9448
10.1016/j.chembiol.2017.05.021 doi
AMP-Activated Protein Kinase Kinases AMP-Activated Protein Kinases--antagonists & inhibitors Allosteric Regulation Binding Sites Catalytic Domain Cell-Free System Enzyme Activation--drug effects HEK293 Cells HeLa Cells Humans Indans--pharmacology Indoles--chemistry Mutagenesis, Site-Directed Niacinamide--analogs & derivatives Phenylurea Compounds--chemistry Phosphorylation--drug effects Protein Isoforms--genetics Protein Serine-Threonine Kinases--metabolism Pyrimidines--pharmacology Sorafenib Sulfonamides--chemistry src-Family Kinases--antagonists & inhibitors