Shchegol'kov, Evgeny V
Synthesis, molecular docking, and biological activity of polyfluoroalkyl dihydroazolo[5,1-c][1,2,4]triazines as selective carboxylesterase inhibitors. [electronic resource]
- Bioorganic & medicinal chemistry 08 2017
- 3997-4007 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3391
10.1016/j.bmc.2017.05.045 doi
Animals
Carboxylesterase--antagonists & inhibitors
Drug Evaluation, Preclinical
Enzyme Inhibitors--chemical synthesis
Humans
Magnetic Resonance Spectroscopy
Molecular Docking Simulation
Structure-Activity Relationship
Triazines--chemical synthesis