Shchegol'kov, Evgeny V

Synthesis, molecular docking, and biological activity of polyfluoroalkyl dihydroazolo[5,1-c][1,2,4]triazines as selective carboxylesterase inhibitors. [electronic resource] - Bioorganic & medicinal chemistry 08 2017 - 3997-4007 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1464-3391

10.1016/j.bmc.2017.05.045 doi


Animals
Carboxylesterase--antagonists & inhibitors
Drug Evaluation, Preclinical
Enzyme Inhibitors--chemical synthesis
Humans
Magnetic Resonance Spectroscopy
Molecular Docking Simulation
Structure-Activity Relationship
Triazines--chemical synthesis