Structure-based virtual screening and optimization of modulators targeting Hsp90-Cdc37 interaction. [electronic resource]
- European journal of medicinal chemistry Aug 2017
- 63-73 p. digital
Publication Type: Journal Article
1768-3254
10.1016/j.ejmech.2017.04.074 doi
Antineoplastic Agents--chemical synthesis Cell Cycle Proteins--antagonists & inhibitors Cell Proliferation--drug effects Chaperonins--antagonists & inhibitors Dose-Response Relationship, Drug Drug Evaluation, Preclinical Drug Screening Assays, Antitumor HSP90 Heat-Shock Proteins--antagonists & inhibitors Humans Molecular Structure Protein Binding--drug effects Small Molecule Libraries--chemical synthesis Structure-Activity Relationship