Oxidized 5-aminosalicylic acid activates Nrf2-HO-1 pathway by covalently binding to Keap1: Implication in anti-inflammatory actions of 5-aminosalicylic acid. [electronic resource]
- Free radical biology & medicine 07 2017
- 715-724 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1873-4596
10.1016/j.freeradbiomed.2017.04.366 doi
Animals Anti-Inflammatory Agents--therapeutic use Colonic Neoplasms--drug therapy HCT116 Cells Heme Oxygenase-1--metabolism Humans Hypochlorous Acid--metabolism Inflammation--drug therapy Inflammatory Bowel Diseases--drug therapy Kelch-Like ECH-Associated Protein 1--metabolism Male Mesalamine--therapeutic use NF-E2-Related Factor 2--metabolism Oxidation-Reduction Protein Binding Rats Rats, Sprague-Dawley