Design, synthesis and SAR of substituted indoles as selective TrkA inhibitors. [electronic resource]
- Bioorganic & medicinal chemistry letters 06 2017
- 2695-2701 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2017.04.045 doi
Dose-Response Relationship, Drug Drug Design Humans Indoles--chemical synthesis Molecular Structure Protein Kinase Inhibitors--chemical synthesis Receptor, trkA--antagonists & inhibitors Structure-Activity Relationship