Hurzy, Danielle M

Design, synthesis and SAR of substituted indoles as selective TrkA inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters 06 2017 - 2695-2701 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2017.04.045 doi


Dose-Response Relationship, Drug
Drug Design
Humans
Indoles--chemical synthesis
Molecular Structure
Protein Kinase Inhibitors--chemical synthesis
Receptor, trkA--antagonists & inhibitors
Structure-Activity Relationship