Insight into the remarkable affinity and selectivity of the aminobenzosuberone scaffold for the M1 aminopeptidases family based on structure analysis. [electronic resource]
- Proteins Aug 2017
- 1413-1421 p. digital
Publication Type: Journal Article
1097-0134
10.1002/prot.25301 doi
Amino Acid Motifs Aminopeptidases--antagonists & inhibitors Anisoles--chemistry Bacterial Proteins--antagonists & inhibitors Catalytic Domain Cloning, Molecular Crystallography, X-Ray Cycloheptanes--chemistry Epoxide Hydrolases--chemistry Escherichia coli--chemistry Gene Expression Humans Kinetics Models, Molecular Protease Inhibitors--chemistry Protein Binding Protein Conformation, alpha-Helical Protein Conformation, beta-Strand Protein Interaction Domains and Motifs Recombinant Proteins--chemistry Sequence Alignment Structural Homology, Protein Substrate Specificity Thermodynamics