Peng, Guanya

Insight into the remarkable affinity and selectivity of the aminobenzosuberone scaffold for the M1 aminopeptidases family based on structure analysis. [electronic resource] - Proteins Aug 2017 - 1413-1421 p. digital

Publication Type: Journal Article

1097-0134

10.1002/prot.25301 doi


Amino Acid Motifs
Aminopeptidases--antagonists & inhibitors
Anisoles--chemistry
Bacterial Proteins--antagonists & inhibitors
Catalytic Domain
Cloning, Molecular
Crystallography, X-Ray
Cycloheptanes--chemistry
Epoxide Hydrolases--chemistry
Escherichia coli--chemistry
Gene Expression
Humans
Kinetics
Models, Molecular
Protease Inhibitors--chemistry
Protein Binding
Protein Conformation, alpha-Helical
Protein Conformation, beta-Strand
Protein Interaction Domains and Motifs
Recombinant Proteins--chemistry
Sequence Alignment
Structural Homology, Protein
Substrate Specificity
Thermodynamics