Chu, Yan-Yan
Rational drug design of indazole-based diarylurea derivatives as anticancer agents. [electronic resource]
- Chemical biology & drug design Oct 2017
- 609-617 p. digital
Publication Type: Journal Article
ISSN: 1747-0285
Standard No.: 10.1111/cbdd.12984 doi
Subjects--Topical Terms: Antineoplastic Agents--chemistry Cell Line, Tumor Cell Proliferation--drug effects Computer-Aided Design Drug Design Drug Screening Assays, Antitumor HCT116 Cells Humans Indazoles--chemistry Molecular Docking Simulation Neoplasms--drug therapy Niacinamide--analogs & derivatives Phenylurea Compounds--pharmacology Proto-Oncogene Proteins c-kit--metabolism Sorafenib Structure-Activity Relationship Urea--analogs & derivatives