Partridge, Katherine M

Discovery and characterization of [(cyclopentyl)ethyl]benzoic acid inhibitors of microsomal prostaglandin E synthase-1. [electronic resource] - Bioorganic & medicinal chemistry letters 03 2017 - 1478-1483 p. digital

Publication Type: Journal Article; Research Support, U.S. Gov't, Non-P.H.S.

1464-3405

10.1016/j.bmcl.2016.11.011 doi


Animals
Benzoates--chemistry
Crystallography, X-Ray
Dogs
Drug Discovery
Microsomes--drug effects
Prostaglandin-E Synthases--antagonists & inhibitors
Rats