TY - GEN AU - Zhao,Peng AU - Nettleton,David O AU - Karki,Rajeshri G AU - Zécri,Frédéric J AU - Liu,Shih-Yuan TI - Medicinal Chemistry Profiling of Monocyclic 1,2-Azaborines SN - 1860-7187 PY - 2017///0627 KW - Administration, Oral KW - Animals KW - Binding Sites KW - Boron Compounds KW - chemistry KW - Chemistry, Pharmaceutical KW - Cyclin-Dependent Kinase 2 KW - antagonists & inhibitors KW - Half-Life KW - Hydrogen Bonding KW - Male KW - Molecular Dynamics Simulation KW - Protein Kinase Inhibitors KW - Protein Structure, Tertiary KW - Rats KW - Rats, Sprague-Dawley KW - Solubility N1 - Publication Type: Journal Article; Research Support, N.I.H., Extramural UR - https://doi.org/10.1002/cmdc.201700047 ER -