Polar aromatic periphery increases agonist potency of spirocyclic free fatty acid receptor (GPR40) agonists inspired by LY2881835. [electronic resource]
- European journal of medicinal chemistry Feb 2017
- 357-368 p. digital
Publication Type: Journal Article
1768-3254
10.1016/j.ejmech.2017.01.005 doi
Animals CHO Cells Caco-2 Cells Cricetinae Cricetulus Drug Design Humans Hypoglycemic Agents--chemical synthesis Molecular Docking Simulation Piperidines--chemistry Protein Conformation Receptors, G-Protein-Coupled--agonists Spiro Compounds--chemical synthesis Structure-Activity Relationship