Krasavin, Mikhail

Polar aromatic periphery increases agonist potency of spirocyclic free fatty acid receptor (GPR40) agonists inspired by LY2881835. [electronic resource] - European journal of medicinal chemistry Feb 2017 - 357-368 p. digital

Publication Type: Journal Article

1768-3254

10.1016/j.ejmech.2017.01.005 doi


Animals
CHO Cells
Caco-2 Cells
Cricetinae
Cricetulus
Drug Design
Humans
Hypoglycemic Agents--chemical synthesis
Molecular Docking Simulation
Piperidines--chemistry
Protein Conformation
Receptors, G-Protein-Coupled--agonists
Spiro Compounds--chemical synthesis
Structure-Activity Relationship