Enhancing the Cell Permeability and Metabolic Stability of Peptidyl Drugs by Reversible Bicyclization. [electronic resource]
- Angewandte Chemie (International ed. in English) 02 2017
- 1525-1529 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
1521-3773
10.1002/anie.201610888 doi
Amino Acid Sequence Cell Membrane Permeability Cell-Penetrating Peptides--chemistry Drug Discovery Drug Stability HeLa Cells Humans I-kappa B Kinase--metabolism Peptides, Cyclic--chemistry Pharmacokinetics Protein Interaction Maps--drug effects Proteolysis Solid-Phase Synthesis Techniques