Li, Ming

The consequence of regional gradients of P-gp and CYP3A4 for drug-drug interactions by P-gp inhibitors and the P-gp/CYP3A4 interplay in the human intestine ex vivo. [electronic resource] - Toxicology in vitro : an international journal published in association with BIBRA Apr 2017 - 26-33 p. digital

Publication Type: Journal Article

1879-3177

10.1016/j.tiv.2016.12.002 doi


ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors
Adult
Aged
Aged, 80 and over
Colon--metabolism
Cyclosporins--pharmacology
Cytochrome P-450 CYP3A--metabolism
Cytochrome P-450 CYP3A Inhibitors--pharmacology
Drug Interactions
Female
Humans
Ileum--metabolism
In Vitro Techniques
Isoquinolines--pharmacology
Jejunum--metabolism
Ketoconazole--pharmacology
Male
Middle Aged
Quinazolines--pharmacology
Quinidine--analogs & derivatives
Verapamil--pharmacology