Novel Hybrid Molecules on the Basis of Steroids and (5Z,9Z)-Tetradeca-5,9-dienoic Acid: Synthesis, Anti-Cancer Studies and Human Topoisomerase I Inhibitory Activity. [electronic resource]
- Anti-cancer agents in medicinal chemistry 2017
- 1126-1135 p. digital
Publication Type: Journal Article
1875-5992
10.2174/1871520616666161207154850 doi
Antineoplastic Agents--chemical synthesis Cell Line, Tumor Cell Proliferation--drug effects Cell Survival--drug effects DNA Topoisomerases, Type I--metabolism Dose-Response Relationship, Drug Drug Screening Assays, Antitumor Fatty Acids, Unsaturated--chemistry Humans Molecular Docking Simulation Molecular Structure Steroids--chemistry Structure-Activity Relationship Topoisomerase I Inhibitors--chemical synthesis