Prostate cancer-associated mutation in SPOP impairs its ability to target Cdc20 for poly-ubiquitination and degradation. [electronic resource]
- Cancer letters 01 2017
- 207-214 p. digital
Publication Type: Journal Article
1872-7980
10.1016/j.canlet.2016.10.021 doi
Antineoplastic Agents--pharmacology Carbamates--pharmacology Cdc20 Proteins--antagonists & inhibitors Cullin Proteins--antagonists & inhibitors Cyclopentanes--pharmacology Diamines--pharmacology Dose-Response Relationship, Drug Drug Resistance, Neoplasm Enzyme Inhibitors--pharmacology HeLa Cells Humans Male Molecular Targeted Therapy Mutation Nuclear Proteins--genetics Prostatic Neoplasms--drug therapy Protein Interaction Domains and Motifs Proteolysis Pyrimidines--pharmacology Repressor Proteins--genetics Time Factors Transfection Ubiquitination