A TPX2 Proteomimetic Has Enhanced Affinity for Aurora-A Due to Hydrocarbon Stapling of a Helix. [electronic resource]
- ACS chemical biology 12 2016
- 3383-3390 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1554-8937
10.1021/acschembio.6b00727 doi
Amino Acid Sequence Aurora Kinase A--chemistry Cell Cycle Proteins--chemistry Crystallography, X-Ray Enzyme Activation Humans Microtubule-Associated Proteins--chemistry Molecular Docking Simulation Nuclear Proteins--chemistry Protein Binding Protein Conformation, alpha-Helical Protein Interaction Maps Thermodynamics