Choi, Hye-Eun

6-(3,4-Dihydro-1H-isoquinoline-2-yl)-N-(6-methoxypyridine-2-yl) nicotinamide-26 (DIMN-26) decreases cell proliferation by induction of apoptosis and downregulation of androgen receptor signaling in human prostate cancer cells. [electronic resource] - Chemico-biological interactions Dec 2016 - 196-207 p. digital

Publication Type: Journal Article

1872-7786

10.1016/j.cbi.2016.10.008 doi


Androgens--pharmacology
Apoptosis--drug effects
Cell Cycle Checkpoints--drug effects
Cell Line, Tumor
Cell Nucleus--drug effects
Cell Proliferation--drug effects
Dihydrotestosterone--pharmacology
Down-Regulation--drug effects
Gene Expression Regulation, Neoplastic--drug effects
Humans
Isoquinolines--chemistry
Male
Prostate-Specific Antigen--genetics
Prostatic Neoplasms--drug therapy
Protein Transport--drug effects
Proto-Oncogene Proteins c-akt--metabolism
RNA, Messenger--genetics
Receptors, Androgen--metabolism
Signal Transduction--drug effects
Transcription, Genetic--drug effects