Blunt, Matthew D
The Dual Syk/JAK Inhibitor Cerdulatinib Antagonizes B-cell Receptor and Microenvironmental Signaling in Chronic Lymphocytic Leukemia. [electronic resource]
- Clinical cancer research : an official journal of the American Association for Cancer Research May 2017
- 2313-2324 p. digital
Publication Type: Journal Article
ISSN: 1557-3265
Standard No.: 10.1158/1078-0432.CCR-16-1662 doi
Subjects--Topical Terms: Adenine--analogs & derivatives Antineoplastic Combined Chemotherapy Protocols--administration & dosage Apoptosis--drug effects B-Lymphocytes--drug effects Bridged Bicyclo Compounds, Heterocyclic--administration & dosage Flow Cytometry Gene Expression Regulation, Neoplastic--drug effects Humans Janus Kinase Inhibitors--administration & dosage Janus Kinases--antagonists & inhibitors Leukemia, Lymphocytic, Chronic, B-Cell--drug therapy Leukocytes, Mononuclear--drug effects Neoplasm Proteins--genetics Piperidines Proto-Oncogene Proteins c-bcr--antagonists & inhibitors Pyrazoles--administration & dosage Pyrimidines--administration & dosage Receptors, Antigen, B-Cell--drug effects Signal Transduction--drug effects Sulfonamides--administration & dosage Sulfones--administration & dosage Syk Kinase--antagonists & inhibitors Tumor Microenvironment--drug effects