First-in-Class Chemical Probes against Poly(ADP-ribose) Glycohydrolase (PARG) Inhibit DNA Repair with Differential Pharmacology to Olaparib. [electronic resource]
- ACS chemical biology 11 2016
- 3179-3190 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1554-8937
10.1021/acschembio.6b00609 doi
DNA Repair Enzyme Inhibitors--pharmacology Glycoside Hydrolases--antagonists & inhibitors HeLa Cells Humans Molecular Probes--chemistry Phthalazines--pharmacology Piperazines--pharmacology Surface Plasmon Resonance