James, Dominic I

First-in-Class Chemical Probes against Poly(ADP-ribose) Glycohydrolase (PARG) Inhibit DNA Repair with Differential Pharmacology to Olaparib. [electronic resource] - ACS chemical biology 11 2016 - 3179-3190 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1554-8937

10.1021/acschembio.6b00609 doi


DNA Repair
Enzyme Inhibitors--pharmacology
Glycoside Hydrolases--antagonists & inhibitors
HeLa Cells
Humans
Molecular Probes--chemistry
Phthalazines--pharmacology
Piperazines--pharmacology
Surface Plasmon Resonance