Discovery of new hit-molecules targeting Plasmodium falciparum through a global SAR study of the 4-substituted-2-trichloromethylquinazoline antiplasmodial scaffold. [electronic resource]
- European journal of medicinal chemistry Jan 2017
- 68-86 p. digital
Publication Type: Journal Article
1768-3254
10.1016/j.ejmech.2016.09.029 doi
Antimalarials--chemical synthesis Cell Survival--drug effects Drug Discovery Hep G2 Cells Humans Plasmodium falciparum--drug effects Quinazolines--chemical synthesis Sensitivity and Specificity Structure-Activity Relationship