Desroches, Justine

Discovery of new hit-molecules targeting Plasmodium falciparum through a global SAR study of the 4-substituted-2-trichloromethylquinazoline antiplasmodial scaffold. [electronic resource] - European journal of medicinal chemistry Jan 2017 - 68-86 p. digital

Publication Type: Journal Article

1768-3254

10.1016/j.ejmech.2016.09.029 doi


Antimalarials--chemical synthesis
Cell Survival--drug effects
Drug Discovery
Hep G2 Cells
Humans
Plasmodium falciparum--drug effects
Quinazolines--chemical synthesis
Sensitivity and Specificity
Structure-Activity Relationship