TY - GEN AU - Adla,Santosh Kumar AU - Slavikova,Barbora AU - Smidkova,Marketa AU - Tloustova,Eva AU - Svoboda,Martin AU - Vyklicky,Vojtech AU - Krausova,Barbora AU - Hubalkova,Pavla AU - Nekardova,Michaela AU - Holubova,Kristina AU - Vales,Karel AU - Budesinsky,Milos AU - Vyklicky,Ladislav AU - Chodounska,Hana AU - Kudova,Eva TI - Physicochemical and biological properties of novel amide-based steroidal inhibitors of NMDA receptors SN - 1878-5867 PY - 2017///0830 KW - Amides KW - Blood-Brain Barrier KW - drug effects KW - Caco-2 Cells KW - Hep G2 Cells KW - Humans KW - Magnetic Resonance Spectroscopy KW - Molecular Structure KW - Neurotransmitter Agents KW - chemistry KW - Reactive Oxygen Species KW - metabolism KW - Receptors, N-Methyl-D-Aspartate KW - antagonists & inhibitors KW - Structure-Activity Relationship N1 - Publication Type: Journal Article; Research Support, Non-U.S. Gov't UR - https://doi.org/10.1016/j.steroids.2016.08.010 ER -